Drug Metabolite

Drug Metabolite

Drug metabolites are created when a drug is metabolized into a different form that still has therapeutic effects. Active metabolites can be produced by drug metabolism redox reactions like heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations. In some rare circumstances, conjugation reactions can also produce an active metabolite. 

Drug Metabolite related products

Structure Cat No. Product Name CAS No. Product Description
V71734 9-Fluorenol (9-Hydroxyfluorene) 1689-64-1 9-Fluorenol (9-Hydroxyfluorene; compound 3) is a DAT (dopamine) inhibitor (antagonist) with IC50 of 9 μM.
V72185 Abiraterone N-oxide 2378463-76-2 Abiraterone N-oxide is the metabolite of Abiraterone.
V72132 Abiraterone sulfate 1993430-25-3 Abiraterone sulfate is the metabolite of Abiraterone.
V30699 Acetaminophen metabolite 3-hydroxy-acetaminophen 37519-14-5 3-hydroxy-acetaminophen is a metabolite of Acetaminophen.
V77781 ACT-606559 ACT-606559 is a new compound with antimalarial activity and is a metabolite of ACT451840.
V72186 Afatinib N-Oxide 2413212-11-8 Afatinib N-Oxide is an impurity during the oxidative degradation of Afatinib dimaleate.
V72165 Ampyrone-d3 (4-Aminoantipyrine-d3) 1329792-51-9 Ampyrone-d3 is the deuterated form of Ampyrone.
V72150 Apalutamide-COOH 1332391-04-4 Apalutamide-COOH is the metabolite of Apalutamide.
V72145 Apovincaminic acid hydrochloride salt 72296-47-0 Apovincaminic acid HCl salt is an orally bioactive and BBB (blood-brain barrier) permeable (penetrable) major bioactive metabolite of Vinpocetine (VP).
V72108 AR-13503 (AR-13324 M1 metabolite) 2309668-15-1 AR-13503 (AR-13324 M1 metabolite) is the hydrolysis metabolite of AR-13324 mesylate.
V69342 AST5902 trimesylate 2929417-90-1 AST5902 trimesylate is the major metabolite of Alflutinib (AST2818) in vivo and in vitro.
V72173 Aszonalenin 81797-27-5 Aszonalenin is a metabolite of Aspergillus zonatus.
V38962 Atorvastatin Epoxy Tetrahydrofuran Impurity 873950-19-7 Atorvastatin Epoxy Tetrahydrofuran Impurity is an oxidative degradation product of Atorvastatin,which is an anti-hyperlipidemic drug and selectiveinhibitor of HMG-CoA reductase.
V69365 AZ7550-d5 2719690-99-8 AZ7550-d5 is the deuterium labelled form of AZ7550.
V32638 Berberrubine chloride 15401-69-1 Berberrubine chloride, a potent metabolite of berberine, reduces symptoms of ulcerative colitis in animal models.
V72270 Bifenazate-diazene 149878-40-0 Bifenazate-diazene is the main degradation product of Bifenazate.
V72290 Captopril EP Impurity B (Captopril EP Impurity B) 80629-35-2 Captopril EP Impurity B is an impurity of Captopril.
V72291 Captopril EP Impurity C (3-Mercaptoisobutyric acid; 3-Mercaptoisobutyric acid) 26473-47-2 Captopril EP Impurity C is an impurity of Captopril.
V72283 Captopril EP Impurity D (3-Bromoisobutyric acid) 56970-78-6 Captopril EP Impurity D is an impurity of Captopril.
V72292 Captopril EP Impurity E (Captopril EP Impurity E) 23500-15-4 Captopril EP Impurity E is an impurity of Captopril.
Contact Us Back to top