AChR Receptor

AChR Receptor

AChR Receptor related products

Structure Cat No. Product Name CAS No. Product Description
V1163 Fesoterodine Fumarate 286930-03-8 Fesoterodine Fumarate (SPM907; Toviaz, SPM-907), the fumarate salt of Fesoterodine which is a prodrug of 5-hydroxymethyl tolterodine, is a muscarinic AChR receptor antagonist that has been approved for treating overactive bladder syndrome.
V1197 Flavoxate HCl (Rec-7-0040; DW61) 3717-88-2 Flavoxate HCl (Rec-7-0040; DW-61; NSC-114649;Rec 7-0040; Rec7-0040; DW61; NSC114649),the hydrochloride salt ofFlavoxate which is a flavanoid,is a muscarinic AChR antagonist with an IC50 of 12.2 μM.
V13604 Galanthamine 357-70-0 Galanthamine is a potent and long-acting AChE inhibitor with IC50 of 0.35 μM, it exhibits 50-fold selectivity against butyryl-cholinesterase.
V1204 Galanthamine HBr 1953-04-4 Galanthamine HBr (Razadyne, Reminyl),the hydrobromide salt ofGalanthamine, is a centrally active and long-acting AChE/acetylcholinesterase inhibitor approved for the treatment of cognitive decline in Alzheimers disease and various other memory impairments.
V1185 Gallamine Triethiodide 65-29-2 Gallamine Triethiodide (Flaxedil; Tricuran; Gallamoni jodidum; Gallaminii iodidum),a non-depolarising muscle relaxant, is a potent and cardioselective cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.
V14212 Glycopyrrolate 596-51-0 Glycopyrrolate (Glycopyrronium bromide, Robinul, Glycopyrrolate bromide,Gastrodyn) is an antispasmodic medication and a muscarinic antagonist used in the treatment of some disorders of the gastrointestinal tract, and to reduce salivation with some anesthetics.
V1201 Hexamethonium Bromide 55-97-0 Hexamethonium Bromide (Vegolysen; Esametina; Simpatoblock),a peripherally-acting and nondepolarizing neuromuscular blocker,is a selective antagonist of neuronal-type nicotinic AChR in ganglia that wasused to treat chronic hypertension.
V1196 Homatropine Bromide (Homatropine hydrobromide) 51-56-9 Homatropine Bromide (Equipin, Isopto Homatropine), the hydrobromide salt of Homatropine, is a potent muscarinic AChR (acetylcholine receptor) antagonist used before eye examinations (i.e. refraction), before and after certain eye surgeries, and for treating certain eye conditions (e.g., uveitis).
V1198 Homatropine Methylbromide (Homatropine methobromide) 80-49-9 Homatropine Methylbromide(Homatropine methobromide),a quaternary ammonium salt of methylhomatropine and a peripherally acting anticholinergic medication, is potent muscarinic AChR antagonist used to treat duodenal or stomach ulcers or intestine problems.
V1178 Ipratropium Bromide (Sch 1000) 22254-24-6 Ipratropium Bromide (Sch 1000; Sch1000; Atrovent, Apovent, Ipraxa, Rinatec) is a potent antagonist of M3 type muscarinic acetylcholine receptors that opens up the medium and large airways in the lungs.
V25120 Isoimperatorin 482-45-1 Isoimperatorin is a COX-2 inhibitor.
V1200 L-Hyoscyamine (Daturine) 101-31-5 L-Hyoscyamine (Daturine), a natural tropane alkaloid and plant toxin, is the the levo-isomer of atropine and is used for controlling symptoms associated with disorders of the gastrointestinal (GI) tract.
V24302 Lobeline hydrochloride (C-07475) 134-63-4 Lobeline hydrochloride,an alkaloid and nonstimulant medication that can alter dopamine uptake in brain,is a novel and potenta nicotinic receptor agonist and VMAT2 ligand, which stimulates dopamine release, and inhibits the reuptake of dopamine and serotonin, acting as a mixed agonist-antagonist at nicotinic acetylcholine receptors and antagonist at µ-opioid receptors.
V1165 LY2119620 886047-22-9 LY2119620 (LY 2119620; LY-2119620) is a novel, potent, specific, high-affinity and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors, the so called positive allosteric modulator (PAM).
V1175 Methscopolamine bromide 155-41-9 Methscopolamine bromide [known also as (-)-Scopolamine methyl bromide; Hyoscine methyl bromide], a methylated scopolamine derivative, is a muscarinic acetylcholine receptor antagonist/blocker that was used to treat peptic ulcers by reducing stomach acid secretion.
V1180 Neostigmine Bromide (Eustigmin; Neoserine) 114-80-7 Neostigmine Bromide (Eustigmin bromide; Neoserine bromide) is a reversible acetylcholinesterase inhibitor and a medication used to treat myasthenia gravis, Ogilvie syndrome, and urinary retention without the presence of a blockage.
V7032 Neostigmine methylsulfate 51-60-5 Neostigmine methylsulfateis a parasympathomimetic compound anda reversible acetylcholinesterase inhibitor.
V1166 Nitenpyram 150824-47-8 Nitenpyram (trade names Capstar, Bestguard),an insect neurotoxin of the neonicotinoid class, is a fast and long-acting, and orally bioavailable nicotinic acetylcholine receptor (AchR) agonist with neural signaling-blocking activity.
V4121 Nitrocaramiphen hydrochloride 98636-73-8 Nitrocaramiphen hydrochloride is a M1 muscarinic (mAChR) antagonist which demonstrates71-foldselectivityforM1overM2.
V1190 Orphenadrine Citrate 4682-36-4 Orphenadrine Citrate (BS-5930;BS5930; BS 5930; Disipal), the citrate salt ofOrphenadrine,is anuncompetitiveNMDA receptor antagonist and apotent skeletal muscle relaxant with antispastic and analgesic activities.
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