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V78794
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14-3-3σ/ERα stabilizer-1 |
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14-3-3σ/ERα stabler-1 (Compound 181) is a covalent 14-3-3σ/ERα stabilizer. |
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V10435
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Afimoxifene (4-hydroxytamoxifen) |
68392-35-8 |
Afimoxifene (4-hydroxytamoxifen or (E/Z)-4-hydroxy Tamoxifen),an active metabolite oftamoxifen with both estrogenic and anti-estrogenic effects, is a SERM (selective estrogen receptor modulator). |
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V1746
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Altrenogest (Allyltrenbolone; RU2267) |
850-52-2 |
Altrenogest (also known as Allyltrenbolone; A35957; RU2267; DRC6246; R-2267;A-35957; RU-2267; Allyl trenbolone; REGU-MATE; Regumate)is a progestogen structurally related to veterinary steroid trenbolone. |
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V12318
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Bazedoxifene |
198481-32-2 |
Bazedoxifene (also known as TSE-424; WAY140424), a novel third generation selective estrogen receptor modulator (SERM) withIC50s of 26 and 99 nM for ERα and ERβ, respectively,has been developed to have favorable effects on bone and the lipid profile while minimizing stimulation of uterine or breast tissues. |
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V1734
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Bazedoxifene acetate (TSE-424) |
198481-33-3 |
Bazedoxifene acetate (formerly TSE-424; WAY140424; WAY-140424; TSE424; Viviant), the acetic acid salt form of Bazedoxifene, is a 3rd generation selective estrogen receptor modulator (SERM) withIC50s of 26 and 99 nM for ERα and ERβ, respectively. |
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V1751
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Bazedoxifene HCl |
198480-56-7 |
Bazedoxifene HCl (formerly TSE-424; WAY-140424; WAY140424; TSE424; Viviant),the hydrochloride salt ofBazedoxifene, is a non-steroidal, indole-based and 3rd generationselective estrogen receptor modulator (SERM) with potential antineoplastic activity. |
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V77195
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Bisphenol AF-d4 (BPAF-d4; 4,4'-(Perfluoropropane-2,2-diyl)diphenol-d4) |
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Bisphenol AF-d4 is an isotopically labeled analog of Bisphenol AF. |
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V17164
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BTC (Estrogen receptor modulator 1) |
63676-22-2 |
BTC, formerly known as RALOXIFENE CORE, is a selective andorally active estrogen receptor modulator (SERM) with apIC50of 0.46. |
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V17369
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Chlorotrianisene |
569-57-3 |
Chlorotrianisene is a long-acting, orally bioactive non-steroidal synthetic estrogen that was used for the treatment of menopause, deficiencies in ovary function, and prostate cancer. |
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V1740
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Clomifene citrate (Clomiphene) |
50-41-9 |
Clomifene Citrate (NSC35770;NSC-35770;Omifin; Chloramiphene;Clomide; Clostilbegit;Clomid; Androxal; Dyneric; Gravosan; Klostilbegit; Serophene), the citrate salt ofClomifene, is a potent SERM (selective estrogen receptor modulator) that has been used in the treatment of ovulation induction. |
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V1733
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Dehydroepiandrosterone (DHEA) |
53-43-0 |
Dehydroepiandrosterone (trans-Dehydroandrosterone; DHEA; Prasterone; Psicosterone; EL-10; GL-701; IP-1001;NSC-9896;PB-007; SH-K-04828; Androstenolone; Diandrone) is an endogenous steroidal hormone acting asan androgen receptor antagonist and an estrogen receptor agonist. |
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V1727
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Dienogest (STS-557) |
65928-58-7 |
Dienogest (formerly BAY86-5258; M-18575; MJR-35; ZK-37659; STS-557; Dinagest; Endometrion; Visanne) is a synthetic and orally bioavailable progesterone that was approved for use in contraception and the treatment of endometriosis. |
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V1732
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Diethylstilbestrol (Stilbestrol) |
56-53-1 |
Diethylstilbestrol (also called Stilbestrol; DES; Distilbene)is a synthetic non-steroidal form of estrogen that can be used to prevent miscarriage and other pregnancy complications as well asin the treatment of menopausal and postmenopausal disorders. |
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V10360
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Dydrogesterone |
152-62-5 |
Dydrogesterone is a synthetic progestin. |
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V1728
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Endoxifen HCl |
1032008-74-4 |
Endoxifen HCl (Z-Endoxifen; N-Desmethyl-4-hydroxytamoxifen), the hydrochloride salt of endoxifen which is an active metabolite of Tamoxifen, is a potent and selective estrogen receptor antagonist/SERM with potential anticancer activity. |
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V1745
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Equol |
531-95-3 |
Equol [(-)-Equol, (3S)-Equol, (S)-Equol, AUS 131] is an isoflavandiol estrogen metabolized from daidzein, specifically, it is produced by intestinal bacteria in response to soy isoflavone intake in human. |
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V79338
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ERα degrader 6 |
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ERα degrader 6 (Compound 31q) is an ERα degrader (KI: 75 nM). |
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V78502
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ERα degrader 7 |
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ERα degrader 7 (Compound B1) is a potent ERα degrader with IC50 of 14.6 nM and a DC 50 of 9.7 nM. |
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V1724
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Estradiol (β-Estradiol) |
50-28-2 |
Estradiol (Oestradiol; Estrace; Dihydrofolliculin; β-Estradiol;17β-estradiol, β-Estradiol; E2; 17β-Oestradiol), the 17-beta-isomer of estradiol, is an endogenous/naturally occuring estrogen steroid hormone and a primary female sex hormone that is involved in the regulation of the estrous and menstrual female reproductive cycles. |
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V1750
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Estradiol Cypionate (Depoestradiol) |
313-06-4 |
Estradiol cypionate (Depoestradiol; β-Estradiol 17-cypionate) is the 17 β-cyclopentylpropinate ester of estradiol used in hormone therapy for menopausal symptoms and low estrogen levels in women. |