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GPCR & G Protein
GPCR & G Protein
♦cAMP
(
0
)
Forskolin (Coleonol; Colforsin)
♦Adenosine Receptor
(
0
)
AZD-4635 (HTL1071)
Reversine
CGS 21680 HCl
Istradefylline (KW-6002)
♦Vasopressin Receptor
(
0
)
Conivaptan HCl (YM 087)
Tolvaptan (OPC-41061)
Mozavaptan (OPC-31260)
♦CXCR
(
0
)
Plerixafor 8HCl (AMD3100)
Plerixafor (AMD 3100)
WZ811
♦CaSR
(
0
)
Cinacalcet HCl (AMG-073)
NPS-2143 (SB-262470)
♦PAFR
(
0
)
Ginkgolide B (BN-52021)
NVP-TNKS656
♦CGRP Receptor
(
0
)
MK-3207 HCl
♦LPA Receptor
(
0
)
Ki16425 (Debio 0719)
Ki16198
♦SGLT
(
0
)
Dapagliflozin (BMS-512148)
Canagliflozin (JNJ 28431754)
Empagliflozin (BI 10773)
Sotagliflozin (LX4211)
♦S1P Receptor
(
0
)
Fingolimod (FTY720) HCl
SKI II
PF-543
Siponimod (BAF312)
Opaganib (ABC294640)
Ozanimod (RPC1063)
Siponimod fumarate (BAF312)
♦Endothelin Receptor
(
0
)
Zibotentan (ZD4054)
Bosentan Hydrate (Ro 47-0203)
Macitentan (ACT-064992 D4)
Sitaxentan sodium (Sitaxsentan; IPI 1040)
Ambrisentan (BSF 208075; LU 208075)
Bosentan
BQ-123
♦Cannabinoid Receptor
(
0
)
Rimonabant (SR141716)
AM1241
AM251
Otenabant (CP-945598) HCl
GW842166X
BML-190 (Indomethacin morpholinylamide; IMMA)
Org 27569
♦5-HT Receptor
(
0
)
Clozapine (HF 1854)
Olanzapine (LY170053)
Ketanserin (R41468)
Fluoxetine HCl (LY-110140)
Latrepirdine (Dimebolin) HCl
Tianeptine sodium
RS-127445
PRX-08066 Maleic acid
Vortioxetine (Lu AA21004) HBr
Buspirone HCl (MJ90221) HCl
Vilazodone HCl (EMD 68843; SB659746A)
Prucalopride Succinate (R-108512, R-93877)
Agomelatine (S-20098; BAN, rINN; Valdoxan, Melitor, Thymanax)
Ondansetron (GR 38032; SN 307; GR-C507/75)
Granisetron HCl (BRL 43694A)
Dapoxetine HCl (LY-210448 HCl)
BRL-15572 dihydrochloride
Rizatriptan Benzoate (MK-462 Benzoate)
SB 271046 HCl (SB-271046A)
LY310762
Risperidone (R-64766; Risperdal)
Ziprasidone HCl (CP-88059)
SB 271046 (SB-271046A)
Trazodone HCl (AF-116;, KB-831)
BMY 7378
Sumatriptan Succinate (GR43175)
Zolmitriptan
Clomipramine HCl (G34586)
Aripiprazole (OPC-14597)
Amitriptyline HCl (Elavil)
Serotonin HCl
Mosapride Citrate (TAK-370; AS-4370)
Eletriptan HBr
WAY-100635 Maleate
Ondansetron HCl (GR 38032; SN 307; GR-C507/75)
Lamotrigine (BW430C; LTG)
BRL-54443
Azasetron HCl (Y-25130)
Duloxetine HCl (LY-248686 HCl)
Fluvoxamine maleate (DU23000 maleate)
Mirtazapine (Org3770; 6-Azamianserin)
SB269970 HCl (SB-269970A)
Intepirdine (SB-742457; GSK-742457; RVT-101)
Blonanserin (AD-5423)
Palonosetron HCl (RS25233-197; Aloxi)
Atomoxetine HCl (Tomoxetine; LY 139603)
Venlafaxine HCl (Wy 45030 HCl)
Urapidil HCl
VUF 10166
Almotriptan Malate (LAS 31416)
Naratriptan HCl (GR-85548A HCl)
Sertraline HCl
Escitalopram Oxalate (Citalopram oxalate)
Loxapine Succinate
Lorcaserin HCl
Desvenlafaxine Succinate (WY 45233; O-Desmethylvenlafaxine)
Desvenlafaxine (WY 45233; O-Desmethylvenlafaxine)
Tropisetron HCl (SDZ-ICS-930 HCl)
Prucalopride (R-108512, R-93877)
Iloperidone (HP-873)
PRX-08066
Vortioxetine lactate
SB269970 (SB-269970A)
♦ Adrenergic Receptor
(
0
)
Piperoxan hydrochloride (Benodaine hydrochloride)
Xylazine HCl (BAY 1470 HCl)
Salbutamol Sulfate (AH-3365; Albuterol)
Doxazosin Mesylate (UK 33274 mesylate)
Asenapine maleate (Org 5222 maleate)
Mirabegron (YM178)
Alfuzosin HCl (SL 77499-10 HCl)
Indacaterol Maleate (QAB149)
Salmeterol Xinafoate (GR 33343X xinafoate)
Labetalol HCl (AH-5158 HCl; Sch-15719W)
Bambuterol HCl (KWD-2183 HCl)
Carteolol HCl (OPC-1085 HCl)
Brimonidine Tartrate (UK 14304; AGN190342)
Betaxolol HCl (SL75212)
Sotalol HCl (MJ 1999)
Detomidine HCl (MPV 253; MPV253)
Acebutolol HCl
Tizanidine HCl (BRN 0618691; AB 021)
Silodosin (KAD 3213; KMD 3213)
Nebivolol (R 065824)
Naftopidil
Clonidine HCl
Oxymetazoline HCl
Maprotiline HCl
Naphazoline HCl
Ritodrine HCl (DU21220 HCl)
Isoprenaline HCl (Isoproterenol HCl)
Carvedilol (BM14190; SKF105517)
DL-Adrenaline
Noradrenaline bitartrate monohydrate
Terbutaline Sulfate
Timolol Maleate (L-714,465 Maleate; MK 950)
Xylometazoline HCl
Clorprenaline HCl
Yohimbine HCl
Synephrine
Epinephrine bitartrate
Phenylephrine HCl
Bisoprolol fumarate
Epinephrine HCl
Formoterol Hemifumarate
Methyldopa (MK-351)
L-Adrenaline
Prazosin HCl
Droxidopa (L-DOPS; SM5688))
Synephrine HCl
Phentolamine Mesylate
Medetomidine HCl (MPV-785)
Ivabradine HCl (Procoralan)
Dexmedetomidine HCl [(S)-Medetomidine]
Cisatracurium Besylate (51W89)
Phenoxybenzamine HCl
Dexmedetomidine
Terazosin HCl dihydrate
Adrenalone HCl
Betaxolol (SL75212)
Tetrahydrozoline HCl (Tetryzoline)
Guanabenz Acetate (BR-750; Wy8678 acetate)
Propranolol HCl (AY64043, ICI45520, NCS91523)
Metoprolol Tartrate
Esmolol HCl
Tolazoline HCl
Scopine
Naftopidil 2HCl
Levobetaxolol HCl (AL-1577A)
♦Histamine Receptor
(
0
)
Clemastine Fumarate (HS592; Meclastine)
Loratadine (Loratidine; SCH 29851)
Azelastine HCl (Allergodil)
Mianserin HCl (ORG GB-94 HCl)
Ranitidine HCl
Bepotastine Besilate (Bepreve)
Ebastine (LAS-W 090; RP64305)
Epinastine HCl (WAL801)
Lidocaine (Lignocaine)
Meclizine 2HCl
Fexofenadine HCl
Cetirizine DiHCl (P071)
Nizatidine
Cimetidine
Diphenhydramine HCl
Olopatadine HCl (ALO4943A; KW4679)
Famotidine (MK208)
Histamine 2HCl (Ergamine)
Levodropropizine (DF-526)
Buclizine HCl (UCB-4445)
Histamine Phosphate
Doxylamine Succinate
Roxatidine acetate HCl (HOE 760)
Ciproxifan (FUB-359)
Brompheniramine maleate
Tetrandrine (NSC-77037)
Ketotifen Fumarate (HC 20511)
Mizolastine (SL 850324)
Lafutidine (FRG-8813)
Betahistine 2HCl
Tripelennamine HCl
Azatadine dimaleate
JNJ-7777120
Chlorpheniramine Maleate
Pemirolast potassium (TWT-8152; BMY 26517)
Desloratadine (Sch34117)
Hydroxyzine 2HCl
Cyclizine 2HCl
Rupatadine Fumarate (UR-12592)
Cyproheptadine HCl
Ibipinabant
♦Dopamine Receptor
(
0
)
PD 128907 HCl
Tetracaine HCl
Benztropine mesylate
Chlorpromazine HCl
Amfebutamone HCl
SKF38393 HCl
Levodopa (L-DOPA)
Rotigotine (N-0437; N-0923)
Metoclopramide HCl
Alizapride HCl
Phenothiazine (NSC2037; ENT38)
Amantadine HCl
Paliperidone
Pramipexole 2HCl Monohydrate
Domperidone (R33812)
Nilvadipine (ARC029; FR34235; FK-235)
Rotundine
Ropinirole HCl
Lurasidone HCl (SM-13496)
Levosulpiride (RV-12309)
Pergolide Mesylate (LY127809)
Dopamine HCl
Penfluridol (R-16341)
Amisulpride (DAN 2163)
SCH-23390 maleate
MPTP hydrochloride
Perphenazine
Prochlorperazine dimaleate salt
♦ Opioid Receptor
(
0
)
Loperamide HCl (R-18553)
Nitrendipine (BAY-E-5009)
JTC-801 HCl
ADL5859 HCl
Lomerizine HCl (KB-2796)
Racecadotril (acetorphan)
(+)-Matrine (Vegard)
Meptazinol HCl
Trimebutine
♦Hedgehog/Smoothened ROCK
(
0
)
Vismodegib (GDC-0449)
Cyclopamine (11-Deoxojervine)
LDE225 (NVP-LDE225,Erismodegib)
Taladegib (LY2940680)
Purmorphamine
PF-5274857
GANT61
Smoothened Agonist (SAG)
Glasdegib (PF-04449913)
SANT-1
BMS-833923 (XL-139)
♦OX Receptor
(
0
)
Suvorexant (MK-4305)
SB408124
Almorexant HCl (ACT 078573)
SB-334867 HCl
Almorexant (ACT 078573)
SB-334867
SB408124 HCl
♦MT Receptor
(
0
)
Ramelteon (TAK-375)
Melatonin
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