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GPCR & G Protein
GPCR & G Protein
♦cAMP
(
0
)
Forskolin (Coleonol; Colforsin)
HJC0350
PACAP 1-27
PACAP 1-38
PACAP 6-38
ESI-05 (NSC 116966)
ST034307
HJC0197
♦Adenosine Receptor
(
0
)
Imaradenant (AZD-4635; HTL1071)
Reversine
CGS 21680 HCl
Istradefylline (KW-6002)
NBMPR
1146188-19-3
SCH-58261
Proxyphylline
Acefylline
A2A receptor antagonist 1
Ciforadenant (CPI-444; V81444)
BAY-545
VIPADENANT
Preladenant (MK-3814; SCH420814)
Capadenoson
Regadenoson (CVT-3146)
Adenosine
ZM241385
Etrumadenant (AB928)
MRS1754
Nicergoline
Idazoxan HCl
Bopindolol Malonate
Norepinephrine (Levarterenol; L-Noradrenaline)
Norepinephrine bitartrate monohydrate
Olodaterol
SR 59230A HCl
Sulmazole
Taminadenant
Terbutaline
Todralazine hydrochloride
Tozadenant
XAC 3HCL
Namodenoson (2 Cl-IB-MECA; CF102)
Metipranolol hydrochloride
Piclidenoson (CF-101)
5'-N-Ethylcarboxamidoadenosine
DPCPX
♦Vasopressin Receptor
(
0
)
Conivaptan HCl (YM 087)
Tolvaptan (OPC-41061)
Mozavaptan (OPC-31260)
Lixivaptan
Balovaptan
Terlipressin acetate
Fuscoside (OPC-21268)
Terlipressin
♦CXCR
(
0
)
Plerixafor 8HCl (AMD3100)
Plerixafor (AMD 3100)
WZ811
SB225002
AMG 487
ATI-2341
AMD 3465 hexahydrobromide
AZD5069
SX-682
Mavorixafor (AMD-070)
CXCR2-IN-1
Navarixin
Reparixin L-lysine salt
Reparixin
SCH 563705
Danirixin
SRT3190
SRT3109
AZD8797
AMD 3465
LIT-927
LY-2510924
Burixafor HBr
NBI-74330
Balixafortide (POL6326)
PS372424 HCl
IT1t dihydrochloride
MSX-122
ML-339
MSX-130
MSX-127 (NSC-23026)
UNBS5162
USL311
VUF11207 fumarate
NUCC-390 diHCl
♦CaSR
(
0
)
Strontium Ranelate (S12911; Distrontium renelate)
Cinacalcet HCl (AMG-073)
NPS-2143 (SB-262470)
Cinacalcet (AMG-073)
ETELCALCETIDE
ETELCALCETIDE HCL
Tecalcet HCl (KRN568; NPS-R568; R568)
NPS-2143 hydrochloride (SB-262470A)
♦PAFR
(
0
)
Ginkgolide B (BN-52021)
NVP-TNKS656
♦CGRP Receptor
(
0
)
MK-3207 HCl
GRA Ex-25
Rimegepant (BMS927711)
MK-3207
UBROGEPANT
Calcitonin salmon
♦LPA Receptor
(
0
)
Ki16425 (Debio 0719)
Ki16198
♦SGLT
(
0
)
Dapagliflozin (BMS-512148)
Canagliflozin (JNJ 28431754)
Empagliflozin (BI 10773)
Sotagliflozin (LX4211)
Phloretin
Phlorizin (Floridzin; NSC 2833)
Bexagliflozin
Dapagliflozin ((2S)-1,2-propanediol hydrate)
♦S1P Receptor
(
0
)
Fingolimod (FTY720) HCl
SKI II
PF-543
Siponimod (BAF312)
Opaganib (ABC294640)
Ozanimod (RPC1063)
PF-429242
CAY10444
Phorbol 12-myristate 13-acetate (PMA)
Siponimod fumarate (BAF312)
Ponesimod
JTE-013 HCl
♦Endothelin Receptor
(
0
)
Zibotentan (ZD4054)
Bosentan Hydrate (Ro 47-0203)
Macitentan (ACT-064992 D4)
Sitaxentan sodium (Sitaxsentan; IPI 1040)
Ambrisentan (BSF 208075; LU 208075)
Bosentan
BQ-123
RO 46-8443
Atrasentan
Atrasentan HCl
RO462005
Macitentan n-butyl analogue
Endothelin 1 swine, human
♦Cannabinoid Receptor
(
0
)
Rimonabant (SR141716)
AM1241
AM251
Otenabant (CP-945598) HCl
GW842166X
BML-190 (Indomethacin morpholinylamide; IMMA)
Org 27569
WIN 55,212-2 Mesylate
RTICBM-189
JD5037
CB1-IN-1 (DBPR211)
Bay 59-3074
BAY-38-7271
Rimonabant HCl (SR141716)
LY2828360
TARANABANT
Linoleylethanolamide
2-Arachidonoylglycerol
AZD-1940
Anandamide
SR144528
Iodopravadoline (AM630)
Otenabant (CP-945598)
N-Arachidonyldopamine
♦5-HT Receptor
(
0
)
Clozapine (HF 1854)
Olanzapine (LY170053)
Ketanserin (R41468)
Fluoxetine HCl (LY-110140)
Latrepirdine (Dimebolin) HCl
Tianeptine sodium
RS-127445
PRX-08066 Maleic acid
Vortioxetine (Lu AA21004) HBr
Buspirone HCl (MJ90221) HCl
Vilazodone HCl (EMD 68843; SB659746A)
Prucalopride Succinate (R-108512, R-93877)
Agomelatine (S-20098; BAN, rINN; Valdoxan, Melitor, Thymanax)
Ondansetron (GR 38032; SN 307; GR-C507/75)
Granisetron HCl (BRL 43694A)
Dapoxetine HCl (LY-210448 HCl)
BRL-15572 dihydrochloride
Rizatriptan Benzoate (MK-462 Benzoate)
SB 271046 HCl (SB-271046A)
LY310762
Risperidone (R-64766; Risperdal)
Ziprasidone HCl (CP-88059)
SB 271046 (SB-271046A)
Trazodone HCl (AF-116;, KB-831)
BMY 7378
Sumatriptan Succinate (GR43175)
Zolmitriptan
Clomipramine HCl (G34586)
Aripiprazole (OPC-14597)
Amitriptyline HCl (Elavil)
Serotonin HCl
Mosapride Citrate (TAK-370; AS-4370)
Eletriptan HBr
WAY-100635 Maleate
Ondansetron HCl (GR 38032; SN 307; GR-C507/75)
Lamotrigine (BW430C; LTG)
BRL-54443
Azasetron HCl (Y-25130)
Duloxetine HCl (LY-248686 HCl)
Fluvoxamine maleate (DU23000 maleate)
Mirtazapine (Org3770; 6-Azamianserin)
SB269970 HCl (SB-269970A)
Intepirdine (SB-742457; GSK-742457; RVT-101)
Blonanserin (AD-5423)
Palonosetron HCl (RS25233-197; Aloxi)
Atomoxetine HCl (Tomoxetine; LY 139603)
Venlafaxine HCl (Wy 45030 HCl)
Urapidil HCl
VUF 10166
Almotriptan Malate (LAS 31416)
Naratriptan HCl (GR-85548A HCl)
Sertraline HCl
Escitalopram Oxalate (Citalopram oxalate)
Loxapine Succinate
Lorcaserin HCl
Desvenlafaxine Succinate (WY 45233; O-Desmethylvenlafaxine)
Desvenlafaxine (WY 45233; O-Desmethylvenlafaxine)
Tropisetron HCl (SDZ-ICS-930 HCl)
Prucalopride (R-108512, R-93877)
Iloperidone (HP-873)
Quetiapine Fumarate (ICI 204636))
Cyclobenzaprine HCl (MK-130)
Flopropione
SEP-363856 HCl (Ulotaront)
Puerarin (Kakonein)
BRL15572 free base
PRX-08066
Vortioxetine lactate
SB269970 (SB-269970A)
8-OH-DPAT
AVN-492
GSK163090
Lu AE58054 hydrochloride
Pardoprunox HCI
TG6-10-1
Ocaperidone (R79598)
Lu AE58054 (Idalopirdine)
LP-211
Pimavanserin
Pimavanserin tartrate
F13714 fumarate
Intepirdine HCl (SB-742457; GSK-742457; RVT-101)
Pardoprunox
Palonosetron
(R,R)-Palonosetron Hydrochloride
LASMIDITAN (COL 144, LY 573144)
Frovatriptan Succinate
Lumateperone tosylate
MK 0893
Vortioxetine (AA21004)
SB 242084 HCl
CP-809101 HCl
SB-399885 HCl
Piboserod
Roluperidone
LY-344864 HCl
Eltoprazine HCl
Pindolol (LB-46)
Sertindole
Ramosetron hydrochloride
Citalopram Hydrobromide (Lu 10-171)
WAY-181187 (SAX-187)
Quetiapine
Aripiprazole monohydrate (OPC14597)
Asenapine (Org 5222)
Cisapride
Ketanserin tartrate
Risperidone Mesylate
Dolasetron (MDL-73147)
Dihydroergotamine Mesylate (DHE; Migranal)
Duloxetine ((S)-Duloxetine; LY248686)
Cyamemazine
Cyproheptadine HCl hydrate
Eptapirone(F11440)
Eucalyptol
Fananserin
Ziprasidone free base
GR 127935 HCl
Lurasidone
Lumateperone toluenesulfonic acid (PTSA salt)
Methotrimeprazine
Metoclopramide hydrochloride hydrate
Ziprasidone HCl hydrate
Zotepine
NLX-101 (F-15599)
PF-04995274
Volinanserin
YL-0919
Ansofaxine hydrochloride ( LY03005; LPM570065)
Tropisetron (SDZ-ICS-930)
Tandospirone (SM3997)
Risperidone hydrochloride
Geissoschizine methyl ether
LY334370
Vilazodone (EMD 68843)
Asenapine HCl (Org 5222 HCl)
Alprenolol
LY 344864
Tandospirone citrate (SM 3997)
Aripiprazole D8
♦ Adrenergic Receptor
(
0
)
Piperoxan hydrochloride (Benodaine hydrochloride)
Xylazine HCl (BAY 1470 HCl)
Salbutamol Sulfate (AH-3365; Albuterol)
Doxazosin Mesylate (UK 33274 mesylate)
Asenapine maleate (Org 5222 maleate)
Mirabegron (YM178)
Alfuzosin HCl (SL 77499-10 HCl)
Indacaterol Maleate (QAB149)
Salmeterol Xinafoate (GR 33343X xinafoate)
Labetalol HCl (AH-5158 HCl; Sch-15719W)
Bambuterol HCl (KWD-2183 HCl)
Carteolol HCl (OPC-1085 HCl)
Brimonidine Tartrate (UK 14304; AGN190342)
Betaxolol HCl (SL75212)
Sotalol HCl (MJ 1999)
Detomidine HCl (MPV 253; MPV253)
Acebutolol HCl
Tizanidine HCl (BRN 0618691; AB 021)
Silodosin (KAD 3213; KMD 3213)
Nebivolol (R 065824)
Naftopidil
Clonidine HCl
Oxymetazoline HCl
Maprotiline HCl
Naphazoline HCl
Ritodrine HCl (DU21220 HCl)
Isoprenaline HCl (Isoproterenol HCl)
Carvedilol (BM14190; SKF105517)
DL-Adrenaline
Noradrenaline bitartrate monohydrate
Terbutaline Sulfate
Timolol Maleate (L-714,465 Maleate; MK 950)
Xylometazoline HCl
Clorprenaline HCl
Yohimbine HCl
Synephrine
Epinephrine bitartrate
Phenylephrine HCl
Bisoprolol fumarate
Epinephrine HCl
Formoterol Hemifumarate
Methyldopa (MK-351)
L-Adrenaline
Prazosin HCl
Droxidopa (L-DOPS; SM5688))
Synephrine HCl
Phentolamine Mesylate
Medetomidine HCl (MPV-785)
Ivabradine HCl (Procoralan)
Dexmedetomidine HCl [(S)-Medetomidine]
Cisatracurium Besylate (51W89)
Phenoxybenzamine HCl
Dexmedetomidine
Terazosin HCl dihydrate
Adrenalone HCl
Betaxolol (SL75212)
Tetrahydrozoline HCl (Tetryzoline)
Guanabenz Acetate (BR-750; Wy8678 acetate)
Propranolol HCl (AY64043, ICI45520, NCS91523)
Metoprolol Tartrate
Esmolol HCl
Tolazoline HCl
Scopine
Naftopidil 2HCl
Levobetaxolol HCl (AL-1577A)
SR-59230A oxalate
Reboxetine mesylate (FCE20124; PNU155950E)
Terazosin HCl
Atipamezole HCl (MPV-1248)
Atipamezole
Tamsulosin HCl
ICI-118551 HCl
Brimonidine (UK 14304; AGN190342)
Batefenterol
Arformoterol tartrate
Arformoterol
Formoterol fumarate dihydrate
Arformoterol Maleate
lofexidine HCl
lofexidine
Tolazoline
ARC-239 dihydrochloride
Amezinium Metilsulfate
Landiolol HCl
Vilanterol trifenatate
Talipexole HCl
Levosalbutamol HCl (Levosalbutamol)
Ritanserin
Bisoprolol
Fenoterol hydrobromide
Fenoterol (Th-1165a; Phenoterol hydrobromide)
Higenamine hydrochloride
Hydrocortisone butyrate
Labetalol (AH-5158; Sch-15719W)
Indacaterol (Onbrez; Arcapta; QAB149)
JP-1302 HCl
Moxisylyte hydrochloride
Nebivolol HCl (R 065824)
Octopamine HCl
Oxprenolol hydrochloride
Xylazine
Metoprolol Succinate
Scopine hydrochloride
Levosalbutamol tartrate (levalbuterol)
Dicentrine
Vilanterol
Lusaperidone
Ivabradine D3 HCl
(S)-Terazosin
Levalbuterol
(R)-Carvedilol
Hydroxybupropion
Arotinolol (Almarl)
♦Histamine Receptor
(
0
)
Clemastine Fumarate (HS592; Meclastine)
Loratadine (Loratidine; SCH 29851)
Azelastine HCl (Allergodil)
Mianserin HCl (ORG GB-94 HCl)
Ranitidine HCl
Bepotastine Besilate (Bepreve)
Ebastine (LAS-W 090; RP64305)
Epinastine HCl (WAL801)
Lidocaine (Lignocaine)
Meclizine 2HCl
Fexofenadine HCl
Cetirizine DiHCl (P071)
Nizatidine
Cimetidine
Diphenhydramine HCl
Olopatadine HCl (ALO4943A; KW4679)
Famotidine (MK208)
Histamine 2HCl (Ergamine)
Levodropropizine (DF-526)
Buclizine HCl (UCB-4445)
Histamine Phosphate
Doxylamine Succinate
Roxatidine acetate HCl (HOE 760)
Ciproxifan (FUB-359)
Brompheniramine maleate
Tetrandrine (NSC-77037)
Ketotifen Fumarate (HC 20511)
Mizolastine (SL 850324)
Lafutidine (FRG-8813)
Betahistine 2HCl
Tripelennamine HCl
Azatadine dimaleate
JNJ-7777120
Chlorpheniramine Maleate
Pemirolast potassium (TWT-8152; BMY 26517)
Desloratadine (Sch34117)
Hydroxyzine 2HCl
Cyclizine 2HCl
Rupatadine Fumarate (UR-12592)
Cyproheptadine HCl
Osthole
Rupatadine
S 38093
Clemizole hydrochloride
GSK189254A
VUF10460
Ibipinabant
Clemizole
Emedastine Difumarate
Emedastine
PITOLISANT
ABT-239
JNJ-39758979
JNJ-31001074
Bavisant dihydrochloride hydrate
SUN-1334H
Bromodiphenhydramine HCl
Astemizole
Decloxizine HCl (UCB-1402; NSC289116)
Chloropyramine
Bepotastine
Diphenhydramine
Psoralenoside
Betahistine mesylate
Conessine
Fexofenadine
Hydroxyzine
Lodoxamide (U42585E)
Lodoxamide Tromethamide
NSC19005
Epinastine (WAL801)
N-Acetylhistamine
Chloropyramine hydrochloride
Fexofenadine D6
Histamine
LML134
♦Dopamine Receptor
(
0
)
PD 128907 HCl
Pramipexole (SND-919)
Tetracaine HCl
Benztropine mesylate
Chlorpromazine HCl
Amfebutamone HCl
SKF38393 HCl
Levodopa (L-DOPA)
Rotigotine (N-0437; N-0923)
Metoclopramide HCl
Alizapride HCl
Phenothiazine (NSC2037; ENT38)
Amantadine HCl
Chlorprothixene
Paliperidone
Pramipexole 2HCl Monohydrate
Domperidone (R33812)
Nilvadipine (ARC029; FR34235; FK-235)
Rotundine
Ropinirole HCl
Lurasidone HCl (SM-13496)
Levosulpiride (RV-12309)
Pergolide Mesylate (LY127809)
Dopamine HCl
Penfluridol (R-16341)
Amisulpride (DAN 2163)
Trimethobenzamide HCl (Ro 2-9578)
SCH-23390 maleate
FAUC-346
GR 103691
MPTP hydrochloride
Perphenazine
Prochlorperazine dimaleate salt
Cariprazine HCl
BP897
Cariprazine
PF-06256142
SB-277011 Dihydrochloride
SCH-23390
PD-168077 maleate
Paliperidone Palmitate
Raclopride tartrate
Dexpramipexole HCl
SKF 82958
Fluoroclebopride
Ropinirole (SKF-101468)
Clozapine N-oxide
Eticlopride HCl
A-381393
ABT-724
Amisulpride HCl
Rotigotine Hydrochloride
Spiperone
Spiperone HCl
Sumanirole maleate
Tavapadon (PF6649751; CVL751)
Nomifensine
Bromocriptine Mesylate (CB-154)
Bromperidol (Impromen; R-11333)
Chlorprothixene HCl
Fenoldopam mesyalte (SKF82526)
Pimozide
(-)-Quinpirole HCl
Droperidol
Nomifensine Maleate
FAUC-365
Fluphenazine HCl
Haloperidol
ITI-722 (Lumateperone)
NGB2904 HCl
Pramipexole 2HCl
Raclopride (FLA-870)
Fenoldopam (SKF 82526)
Tetrahydroberberine
rac-Rotigotine Hydrochloride
ML417
ABT-724 trihydrochloride
♦ Opioid Receptor
(
0
)
Loperamide HCl (R-18553)
Nitrendipine (BAY-E-5009)
JTC-801 HCl
ADL5859 HCl
Lomerizine HCl (KB-2796)
Racecadotril (acetorphan)
(+)-Matrine (Vegard)
Meptazinol HCl
Trimebutine
AR-M 1000390 HCl
CYM51010
(R)-(-)-GR103545 fumarate
SR17018
Cebranopadol ((1α,4α)stereoisomer)
Alvimopan
Alvimopan monohydrate
Alvimopan dihydrate
BAN-ORL-24 HCl
LY2795050
LY2940094
Aticaprant (CERC-501)
PZM21
Asimadoline
SNC80
Difelikefalin
LY-2940094 tartrate
DAMGO TFA
DAMGO
Porcine dynorphin A(1-13)
♦Hedgehog/Smoothened ROCK
(
0
)
Vismodegib (GDC-0449)
Cyclopamine (11-Deoxojervine)
LDE225 (NVP-LDE225,Erismodegib)
Taladegib (LY2940680)
Purmorphamine
PF-5274857
GANT61
Smoothened Agonist (SAG)
Glasdegib (PF-04449913)
SANT-1
BMS-833923 (XL-139)
♦OX Receptor
(
0
)
Suvorexant (MK-4305)
SB408124
Almorexant HCl (ACT 078573)
SB-334867 HCl
IPSU
Almorexant (ACT 078573)
SB-334867
SB408124 HCl
TCS-OX2-29
MK-1064
Orexin 2 Receptor Agonist
TCS 1102
SB-649868
JNJ-10397049
GSK1059865
TCS-OX2-29 HCl
GSK1059865 HCl
MK-6096 (Filorexant)
MK-3697
SB-674042
Lemborexant (E-2006)
Orexin A human, rat, mouse
EMPA
♦MT Receptor
(
0
)
Ramelteon (TAK-375)
Melatonin
♦Guanylate Cyclase
(
0
)
Riociguat (BAY 63-2521)
BAY 41-2272
PLECANATIDE
ODQ
Nelociguat
Vericiguat
Cinaciguat
Cinaciguat HCl
Linaclotide
BAY-41-8543
Ebselen oxide
Lificiguat (YC 1)
LY83583
Methylthioninium chloride hydrate
Plecanatide acetate
♦LPL Receptor
(
0
)
Pluronic F-68
GLPG2938
ONO-7300243
CYM-5541 (ML249)
BMS-986020
GSK2018682
Ceralifimod
Amiselimod HCl
CYM-5442
AM095 sodium
SEW2871
Cenerimod
YUN88562
CYM-50308
Etrasimod
Mocravimod (KRP-203) HCl
AM095 free acid
Lysophosphatidic acid
♦NPY receptor
(
0
)
CGP-71683A HCl
♦Angiotensin Receptor
(
0
)
PD-123319 TFA salt
tranilast
Sparsentan
CGP-42112
Olodanrigan (PD126055; EMA 401)
Tasosartan
Olmesartan (RNH-6270; CS-866)
Angiotensin acetate
AT2 Agonist C21 (M24)
AVE 0991
AVE-0991 sodium
Azilsartan mepixetil
Irbesartan HCl
Eprosartan (SKF-108566J)
Losartan (DUP 89)
Azilsartan medoxomil monopotassium (TAK 491)
Tranilast trans-
Candesartan D4 (CV-11974 D4)
Losartan D4 Carboxylic Acid
Losartan D4
Losartan Carboxylic Acid
♦Free Fatty Acid Receptor
(
0
)
AMG-837 calcium hydrate
GSK137647A
GPR120 Agonist 2
TUG-770
GW1100
Vincamine
Pinocembrin racemate (DL0108)
AR-420626
TUG-891
GPR40/FFAR1 modulator 1
♦GnRH Receptor
(
0
)
ELAGOLIX
Elagolix sodium
Degarelix
Relugolix
Cetrorelix acetate (SB-75)
Abarelix
Alarelin Acetate
Degarelix acetate
Goserelin Acetate
[D-Arg6,Pro9-NEt]Salmon gonadotropin-releasing hormone
♦GPR
(
0
)
ML-191
APD597 (JNJ38431055)
APD 668
DJ-V159
JNJ 63533054
CID-16020046
AF64394
ONC212
CID2440433
FTBMT
GTPL5846
JMS-17-2
LP-471756
ML401
MBX-2982 (SAR260093)
ML-193
NIBR-189
AR 231453
DC260126
NE 52-QQ57
ML 145
♦Leukotriene Receptor
(
0
)
Olsalazine Sodium (CJ-91B)
MK-571 Sodium (L-660711)
MONTELUKAST SODIUM (MK0476)
Pranlukast
CP105696
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Montelukast Dicyclohexylamine
♦mAChR
(
0
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VU0238441
TBPB
VU0357017 HCI
Pirmenol (Cl-845)
Umeclidinium bromide
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BQCA
MK-7622
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Xanomeline oxalate
Norclozapine (ACP-104)
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Harmaline
Benzetimide HCl
Biperiden Hydrochloride
Scopolamine HCl
Tiotropium bromide
Tolterodine
DREADD agonist 21
VU0119498
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Mepenzolate Bromide
VU0453595
Bethanechol
Pirmenol hydrochloride
Oxotremorine M iodide
Racanisodamine
Pilocarpine nitrate
mAChR-IN-1
Clozapine N-oxide diHCl
♦Neurotensin Receptor
(
0
)
Talnetant (SB 223412)
LM11A-31 HCl
ML314
AF38469
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