| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V86633 | GPR84 agonist-1 | 489403-70-5 | GPR84 agonist-1 (Compound LY214-5) is a GPR84 agonist with EC50 of 2.479 μM. |
|
V136879 | GPR84 agonist-2 | 3105662-82-3 | GPR84 agonist-2 is a selective GPR84 agonist that is inactive against free fatty acid receptors. |
|
V75420 | GPR84 antagonist 1 | 2762180-28-7 | GPR84 antagonist 1 is a high-affinity, selective competitive antagonist of human GPR84. |
|
V136880 | GPR84 antagonist 10 | 2654791-94-1 | GPR84 antagonist 10 is a potent and orally effective GPR84 antagonist. |
|
V75418 | GPR84 antagonist 2 | 2244269-74-5 | GPR84 antagonist 2 (compound 33) is an orally bioactive, selective GPR84 antagonist (IC50=8.95 nM). |
|
V75421 | GPR84 antagonist 3 | 2815263-05-7 | GPR84 antagonist 3 (compound 42) is a potent GPR84 (G protein-coupled receptor 84) antagonist. |
|
V86632 | GPR84 antagonist 9 | 2654791-96-3 | GPR84 antagonist 9 is an orally active GPR84 antagonist with IC50 of 0.012 μM. |
|
V75423 | GPR88 agonist 2 | 2821859-71-4 | GPR88 agonist 2 (compound 53) is a potent, BBB (blood-brain barrier) permeable (penetrable) GPR88 agonist/activator with EC50 of 14 nM in GPR88 cAMP functional assays. |
|
V85742 | GPR88 agonist 3 | 2963597-44-4 | |
|
V75422 | GPR88-IN-1 | 714265-50-6 | GPR88-IN-1 is a GPR88 inhibitor that may be utilized in the research/study of central diseases. |
|
V1804 | GSK1292263 | 1032823-75-8 | GSK1292263 is a novel and potentGPR119 (G-protein-coupled receptor 119) agonist whichhas potential for the treatment of type 2 diabetes. |
|
V137028 | GW856464 | 851690-21-6 | GW856464 is an antagonist of MCHR1. |
|
V1805 | GW9508 | 885101-89-3 | GW9508 is a novel, potent and selective agonist for FFA1 (fatty acid receptor GPR40) with pEC50 of 7.32, and is 100-fold selective against GPR120, it stimulates insulin secretion in a glucose-sensitive manner. |
|
V137266 | HEP-50768 | 3036387-75-1 | HEP-50768 is an orally effective selective MRGPRX4 (hX4) antagonist. |
|
V70560 | hMCH-1R antagonist 1 | 353487-64-6 | hMCH-1R antagonist 1 (Compound 30) is a potent and specific human melanin concentrating hormone receptor 1 (hMCHR1) antagonist (inhibitor) with a KB of 3.6 nM. |
|
V138336 | K-833 | 2639936-77-7 | K-833 is a GPR119 agonist with EC50 values of 39.8 nM in humans, 100 nM in mice, 75.4 nM in rats, and 12.6 nM in dogs. |
|
V70310 | L-α-lysophosphatidylinositol (Soy) (sodium) | 796963-91-2 | L-α-lysophosphatidylinositol Soy sodium is the endogenous ligand of GPR55. |
|
V139515 | MCH-1 antagonist 2 | 345-24-4 | MCH-1 antagonist 2 is a melanin-concentrating hormone-1 (MCH1) receptor-selective 4-arylpiperidine. |
|
V140399 | MrgprX2 antagonist-10 | 3116848-78-0 | MrgprX2 antagonist-10 is a MrgprX2 antagonist with an IC50 of less than 100 nM. |
|
V140400 | MrgprX2 antagonist-11 | 3116847-13-0 | MrgprX2 antagonist-11 is a MrgprX2 antagonist with an IC50 of less than 100 nM. |
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